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An Innovation 10 Years in the Making: The Stories in the Pages of ACS  Medicinal Chemistry Letters | ACS Medicinal Chemistry Letters
An Innovation 10 Years in the Making: The Stories in the Pages of ACS Medicinal Chemistry Letters | ACS Medicinal Chemistry Letters

Expanding the Medicinal Chemist Toolbox: Comparing Seven C(sp2)–C(sp3)  Cross-Coupling Methods by Library Synthesis | ACS Medicinal Chemistry  Letters
Expanding the Medicinal Chemist Toolbox: Comparing Seven C(sp2)–C(sp3) Cross-Coupling Methods by Library Synthesis | ACS Medicinal Chemistry Letters

Novel Reagent Space: Identifying Unorderable but Readily Synthesizable  Building Blocks | ACS Medicinal Chemistry Letters
Novel Reagent Space: Identifying Unorderable but Readily Synthesizable Building Blocks | ACS Medicinal Chemistry Letters

Relevance of the Trillion-Sized Chemical Space “eXplore” as a Source for  Drug Discovery | ACS Medicinal Chemistry Letters
Relevance of the Trillion-Sized Chemical Space “eXplore” as a Source for Drug Discovery | ACS Medicinal Chemistry Letters

Discovery of Potent Deuterated Compounds as Potential KRASG12D Inhibitors  in Cancer Therapy | ACS Medicinal Chemistry Letters
Discovery of Potent Deuterated Compounds as Potential KRASG12D Inhibitors in Cancer Therapy | ACS Medicinal Chemistry Letters

Systematic Study of Effects of Structural Modifications on the Aqueous  Solubility of Drug-like Molecules | ACS Medicinal Chemistry Letters
Systematic Study of Effects of Structural Modifications on the Aqueous Solubility of Drug-like Molecules | ACS Medicinal Chemistry Letters

ACS Medicinal Chemistry Letters | Vol 11, No 11
ACS Medicinal Chemistry Letters | Vol 11, No 11

ACS Medicinal Chemistry Letters: Volume 11, Issue 5
ACS Medicinal Chemistry Letters: Volume 11, Issue 5

Addition of Fluorine and a Late-Stage Functionalization (LSF) of the Oral  SERD AZD9833 | ACS Medicinal Chemistry Letters
Addition of Fluorine and a Late-Stage Functionalization (LSF) of the Oral SERD AZD9833 | ACS Medicinal Chemistry Letters

Discovery and Development of Cyclic Peptide Inhibitors of CIB1 | ACS  Medicinal Chemistry Letters
Discovery and Development of Cyclic Peptide Inhibitors of CIB1 | ACS Medicinal Chemistry Letters

Discovery of Spiro-azaindoline Inhibitors of Hematopoietic Progenitor  Kinase 1 (HPK1) | ACS Medicinal Chemistry Letters
Discovery of Spiro-azaindoline Inhibitors of Hematopoietic Progenitor Kinase 1 (HPK1) | ACS Medicinal Chemistry Letters

Design, Synthesis, and Anti-HBV Activity of New Bis(l-amino acid) Ester  Tenofovir Prodrugs | ACS Medicinal Chemistry Letters
Design, Synthesis, and Anti-HBV Activity of New Bis(l-amino acid) Ester Tenofovir Prodrugs | ACS Medicinal Chemistry Letters

Targeted Covalent Inhibition of Plasmodium FK506 Binding Protein 35 | ACS  Medicinal Chemistry Letters
Targeted Covalent Inhibition of Plasmodium FK506 Binding Protein 35 | ACS Medicinal Chemistry Letters

Discovery of a Series of 3-Cinnoline Carboxamides as Orally Bioavailable,  Highly Potent, and Selective ATM Inhibitors | ACS Medicinal Chemistry  Letters
Discovery of a Series of 3-Cinnoline Carboxamides as Orally Bioavailable, Highly Potent, and Selective ATM Inhibitors | ACS Medicinal Chemistry Letters

GSK973 Is an Inhibitor of the Second Bromodomains (BD2s) of the Bromodomain  and Extra-Terminal (BET) Family | ACS Medicinal Chemistry Letters
GSK973 Is an Inhibitor of the Second Bromodomains (BD2s) of the Bromodomain and Extra-Terminal (BET) Family | ACS Medicinal Chemistry Letters

Structural and Functional Characterization of Indane-Core CD4-Mimetic  Compounds Substituted with Heterocyclic Amines | ACS Medicinal Chemistry  Letters
Structural and Functional Characterization of Indane-Core CD4-Mimetic Compounds Substituted with Heterocyclic Amines | ACS Medicinal Chemistry Letters

Readily Accessible High-Throughput Experimentation: A General Protocol for  the Preparation of ChemBeads and EnzyBeads | ACS Medicinal Chemistry Letters
Readily Accessible High-Throughput Experimentation: A General Protocol for the Preparation of ChemBeads and EnzyBeads | ACS Medicinal Chemistry Letters

Phenyl Dihydrouracil: An Alternative Cereblon Binder for PROTAC Design | ACS  Medicinal Chemistry Letters
Phenyl Dihydrouracil: An Alternative Cereblon Binder for PROTAC Design | ACS Medicinal Chemistry Letters

Massively Parallel Optimization of the Linker Domain in Small Molecule  Dimers Targeting a Toxic r(CUG) Repeat Expansion | ACS Medicinal Chemistry  Letters
Massively Parallel Optimization of the Linker Domain in Small Molecule Dimers Targeting a Toxic r(CUG) Repeat Expansion | ACS Medicinal Chemistry Letters

Scaffold-Hopping of Aurones: 2-Arylideneimidazo[1,2-a]pyridinones as  Topoisomerase IIα-Inhibiting Anticancer Agents | ACS Medicinal Chemistry  Letters
Scaffold-Hopping of Aurones: 2-Arylideneimidazo[1,2-a]pyridinones as Topoisomerase IIα-Inhibiting Anticancer Agents | ACS Medicinal Chemistry Letters

Discovery of N-(1-Acryloylazetidin-3-yl)-2-(1H-indol-1-yl)acetamides as  Covalent Inhibitors of KRASG12C | ACS Medicinal Chemistry Letters
Discovery of N-(1-Acryloylazetidin-3-yl)-2-(1H-indol-1-yl)acetamides as Covalent Inhibitors of KRASG12C | ACS Medicinal Chemistry Letters

Artificial Intelligence in Drug Design—The Storm Before the Calm? | ACS  Medicinal Chemistry Letters
Artificial Intelligence in Drug Design—The Storm Before the Calm? | ACS Medicinal Chemistry Letters

Identification of New Small-Molecule Inducers of Estrogen-related Receptor  α (ERRα) Degradation | ACS Medicinal Chemistry Letters
Identification of New Small-Molecule Inducers of Estrogen-related Receptor α (ERRα) Degradation | ACS Medicinal Chemistry Letters